News of 2024-11 Nov

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News of November 2024.

ZINC-22 3D database updates

  • zinc-22j now has about 220M new 3D molecules. Growing.
  • zinc-22j H04-H18 complete. H19 is 50%. H20 3%. H21 0%
  • zinc-22y is now up to 1.8 billion. Growing.
  • zinc-22y H04-H21 complete. H22 96%. H23 50%. H24 10%.
  • zinc-22n and zinc-22x - some incremental updates and fixes.
  • macrocycles zinc-22w,e,f are subject to rapid change.
  • strategy: we will get zinc-22y complete to H24, then zinc-22j to H24.
  • strategy: we will finish installing everything built H25-H29.
  • strategy: Then we will do a delta and build the balance as zinc-22y.

Selective syncing to Wynton

  • formerly, we did not sync H26 and above. Now we do.
  • as of 11/21/2024 the following no longer exist on Wynton
  • update: as of 12/15/24 it is now just :
  • zinc-22n/H??/*/[k-z]
  • zinc-22x/H??/*/[k-z]
  • that's right, we are down to 10/26 (38.5%) on Wynton for the "x" and "n" layers.
  • the balance of which k-z can be docked on gimel or aws.
  • to be clear: only the n and x layers are affected.
  • all other layers and tranches are 100% present on Wynton.
  • note, we are still expecting (12/15/24) 312-50 = 262 TB of disk space.
  • Even when this arrives we will not be able to host all of ZINC-22 on Wynton.
  • To host all of ZINC-22 3D on Wynton that is built as of today, I estimate we need to spend $100,000+

Release of Iron-24

We are enumerating the Hartenfeller/Enamine/public reactions. This and the Ir database below, are the Enumerated databases enabled by the Chemistry Commons

We are also enumerating, using the same reactions, the following:

Release of Iridium-24

We are enumerating the bespoke libraries (Ellman, Young, others)

Other news

  • informer set /zinc-22a/ was updated in August 2024. Working on another update.
  • tldr-dev.docking.org and tldr.docking.org will be merged in December 2024.
  • we have started using discord to discuss